Chem Biol Drug Des 76:77–81. doi:10.1111/j.1747-0285.2010.00977.x PubMedCrossRef Flentke GR, Munoz E, Huber BT, Plaut AG, Kettner CA, Bachovchin WW (1991) Inhibition of dipeptidyl aminopeptidase IV (DP-IV) by Xaa-boroPro dipeptides and use of these inhibitors to examine the role of DP-IV in T-cell function. Proc Natl Acad Sci USA 88:1556–1559PubMedCrossRef Fujita T, Kumamoto E
(2006) Inhibition by endomorphin-1 and endomorphin-2 of excitatory Temsirolimus transmission in adult rat substantia gelatinosa neurons. Neuroscience 139:1095–1105. doi:10.1016/j.neuroscience.2006.01.010 PubMedCrossRef Grass S, Xu IS, Wiesenfeld-Hallin Z, Xu X-J (2002) Comparison of the effect of intrathecal endomorphin-1 and endomorphin-2 on spinal cord excitability in rats. Neurosci Lett 324:197–200. selleck screening library doi:10.1016/S0304-3940(02)00201-X PubMedCrossRef Horvath G (2000) Endomorphin-1 and endomorphin-2: pharmacology of the selective endogenous μ-opioid receptor agonist. Pharmacol Ther 88:437–463. doi:10.1016/S0163-7258(00)00100-5 PubMedCrossRef Horvath G, Szikszay M, Tomboly C, Benedek G (1999) Antinociceptive effects of intrathecal endomorphin-1 and -2 in rats. Life Sci 65:2635–2641. doi:10.1016/S0024-3205(99)00532-9 PubMedCrossRef Keresztes A, Borics A, Tóth G (2010) Recent advances in endomorphin engineering. Chem Med Chem. doi:10.1002/cmdc.201000077 Li
J, Wilk E, Wilk S (1995) Aminoacylpyrrolidine-2-nitriles: potent and stable inhibitors of dipeptidyl-peptidase IV (CD 26). Arch Biochem Biophys 323:148–154. https://www.selleckchem.com/products/prt062607-p505-15-hcl.html doi:10.1006/abbi.1995.0020 PubMedCrossRef Mentlein R (1999) Dipeptidyl-peptidase IV (CD26)—role in the inactivation of regulatory peptides. Regul Pept 85:9–24.
doi:10.1016/S0167-0115(99)00089-0 Calpain PubMedCrossRef Narita M, Mizoguchi H, Oji DE, Dun NJ, Hwang BH, Nagase H, Tseng LF (1999) Identification of the G-protein-coupled ORL1 receptor in the mouse spinal cord by [35S]-GTPgammaS binding and immunohistochemistry. Br J Pharmacol 128:1300–1306PubMedCrossRef Peter A, Toth G, Tomboly C, Laus G, Tourwe D (1999) Liquid chromatographic study of the enzymatic degradation of endomorphins, with identification by electrospray ionization mass spectrometry. J Chromatogr A 846:39–48PubMedCrossRef Przewłocki R, Przewłocka B (2001) Opioids in chronic pain. Eur J Pharmacol 429:79–91. doi:10.1016/S0014-2999(01)01308-5 PubMedCrossRef Sakurada C, Sakurada S, Hayashi T, Katsuyama S, Tan-No K, Sakurada T (2003) Degradation of endomorphin-2 at the supraspinal level in mice is initiated by dipeptidyl peptidase IV: an in vitro and in vivo study. Biochem Pharmacol 66:653–661. doi:10.1016/S0006-2952(03)00391-5 PubMedCrossRef Schon E, Born I, Demuth HU, Faust J, Neubert K, Steinmetzer T, Barth A, Ansorge S (1991) Dipeptidyl peptidase IV in the immune system.